HBTU mediated 1-hydroxybenzotriazole (HOBt) conjugate addition: synthesis and stereochemical analysis of β-benzotriazole N-oxide substituted γ-amino acids and hybrid peptides
Author:
Affiliation:
1. Department of Chemistry
2. Indian Institute of Science Education and Research
3. Pune-411 008, India
Abstract
Synthesis and conformational analysis of β-benzotriazole N-oxide (β-BtO) substituted γ-amino acids by direct conjugate addition of HOBt to E-vinylogous γ-amino acids are reported.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2014/OB/C4OB01548G
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