Amino- and chloro-8-hydroxyquinolines and their copper complexes as proteasome inhibitors and antiproliferative agents

Author:

Oliveri Valentina12345ORCID,Lanza Valeria67895ORCID,Milardi Danilo67895ORCID,Viale Maurizio101112135,Maric Irena101112135,Sgarlata Carmelo12345ORCID,Vecchio Graziella12345ORCID

Affiliation:

1. Dipartimento di Scienze Chimiche

2. Università degli Studi di Catania

3. Viale A. Doria 6

4. 95125 Catania

5. Italy

6. Istituto di Biostrutture e Bioimmagini

7. CNR

8. Via P. Gaifami 18

9. 95126 Catania

10. Ospedale Policlinico San Martino

11. U.O.C. Bioterapie

12. Lgo R. Benzi 10

13. 16132, Genova

Abstract

5-Aminomethyl-8-hydroquinoline and its copper(ii) complex look very promising in inhibiting cell growth and proteasome activity.

Funder

Ministero dell'Istruzione, dell'Università e della Ricerca

Publisher

Oxford University Press (OUP)

Subject

Metals and Alloys,Biochemistry,Biomaterials,Biophysics,Chemistry (miscellaneous)

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