Organocatalytic [4+1]-annulation approach for the synthesis of densely functionalized pyrazolidine carboxylates
Author:
Affiliation:
1. Chemical Engineering & Process Development Division
2. CSIR-National Chemical Laboratory
3. Pune
4. India-411008
Abstract
The present protocol provides optically active pyrazolidine carboxylates with derivatizable functional groups in high yields with excellent enantio- and diastereoselectivities.
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA09583B
Reference81 articles.
1. Heterocyclic Compounds as Anti-Inflammatory Agents
2. J. Elguero in Comprehensive Heterocyclic Chemistry, ed. K. T. Potts, Pergamon Press, Oxford, 1984, vol. 5, p. 167
3. Ring-opening cross metathesis of 1,3-cyclopentadiene-heterodienophile cycloadducts to produce cyclic hydrazines and hydroxylamines
4. L. C. Behr , R.Fusco and C. H.Jarboe, in The Chemistry of Heterocyclic Compounds, Pyrazoles, Pyrazolines, Pyrazolidines, Indazoles and Condensed Rings, ed. A. Weissberger, Interscience Publishers, New York, 1967
5. Versatile, Diastereoselective Additions of Silyl Ketene Acetals, Allyl Tributylstannane, and Me3SiCN to N-Acyl Pyrazolines: Asymmetric Synthesis of Densely Functionalized Pyrazolidines
Cited by 6 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Pyrazolidines: synthesis, reactivity, physical and biological properties;Arkivoc;2024-06-25
2. Recent advances in the application of ylide-like species in [4 + 1]-annulation reactions: an updated review;Organic Chemistry Frontiers;2022
3. Diastereoselective Synthesis of Chiral 2,3-Disubstituted Indolines via Formal [3+2]-Cycloaddition of Arynes with γ-Amino-α,β-unsaturated Esters;The Journal of Organic Chemistry;2017-05-22
4. Proline catalyzed enantioselective synthesis of (2 S ,3 S )-3-hydroxypipecolic acid and formal synthesis of (+)-swainsonine;Tetrahedron Letters;2016-05
5. A Concise Enantioselective Synthesis of (+)-L-733,060 and (+)-T-2328 via Sequential Proline Catalysis;Synlett;2016-02-04
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3