Affiliation:
1. Nicolaus Copernicus University in Toruń, Faculty of Chemistry, 7 Gagarin Street, 87-100 Toruń, Poland
Abstract
The direct and highly enantioselective C3-functionalization of the 2,1-benzothiazine 2,2-dioxide skeleton using NHC-catalyzed generation of chiral α,β-unsaturated acylazoliums, showcasing a synthesis pathway with enhanced pharmacological potential.
Publisher
Royal Society of Chemistry (RSC)
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