Dimeric polyphenols to pave the way for new antimalarial drugs

Author:

Degotte Gilles12ORCID,Pendeville Hélène3,Di Chio Carla4,Ettari Roberta4,Pirotte Bernard1ORCID,Frédérich Michel2,Francotte Pierre1

Affiliation:

1. Laboratory of Medicinal Chemistry, CIRM, Department of Pharmacy, University of Liège, Quartier Hôpital – B36 Tower 4, +5, Avenue Hippocrate 15, 4000 Liège, Belgium

2. Laboratory of Pharmacognosy, CIRM, Department of Pharmacy, University of Liège, Quartier Hôpital – B36 Tower 4, +5, Avenue Hippocrate 15, 4000 Liège, Belgium

3. Platform Zebrafish facility & transgenics, GIGA, University of Liège, Quartier Hôpital – B34, +2, Avenue de l'Hôpital 11, 4000 Liège, Belgium

4. Dipartimento di Scienze chimiche, biologiche, farmaceutiche e ambientali, Università degli Studi di Messina, Viale Annunziata, 98168 Messina, Italy

Abstract

A polyphenolic scaffold to develop novel orally active antimalarials against resistant Plasmodium falciparum.

Funder

Fonds Léon Fredericq

Fonds pour la Formation à la Recherche dans l’Industrie et dans l’Agriculture

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Reference70 articles.

1. World Health Organisation , Distribution of Causes of Death Among Children aged < 5 years , https://www.who.int/data/gho/data/indicators/indicator-details/GHO/distribution-of-causes-of-death-among-children-aged-5-years-(-) , (accessed 8 April 2021 )

2. World Health Organization , World malaria report 2021 , 2021

3. Center for Disease Control , Anopheles Mosquitoes, https://www.cdc.gov/malaria/about/biology/index.html#tabs-1-5 , (accessed 27 January 2021)

4. Center for Disease Control , Biology , https://www.cdc.gov/malaria/about/biology/index.html , (accessed 27 January 2021)

5. World Health Organization , Malaria , https://www.who.int/news-room/fact-sheets/detail/malaria , (accessed 8 April 2021)

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