An insight into tetrahydro-β-carboline–tetrazole hybrids: synthesis and bioevaluation as potent antileishmanial agents
Author:
Affiliation:
1. Medicinal and Process Chemistry Division
2. CSIR-Central Drug Research Institute
3. Lucknow-226031
4. India
5. Division of Biochemistry
6. Pharmacokinetics & Metabolism Division
7. Lucknow
Abstract
A series of tetrahydro-β-carboline tetrazole derivatives have been synthesized utilizing the Ugi-tetrazole reaction and were identified as potential antileishmanial chemotypes.
Publisher
Royal Society of Chemistry (RSC)
Subject
Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2017/MD/C7MD00125H
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