Catechols: a new class of carbonic anhydrase inhibitors-Reference-Cited by-同舟云学术

Catechols: a new class of carbonic anhydrase inhibitors

Published:2020 Issue:85 Volume:56 Page:13033-13036
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

D'Ambrosio Katia¹²³^ORCID,Carradori Simone⁴⁵⁶³^ORCID,Cesa Stefania⁷⁸⁹³^ORCID,Angeli Andrea¹⁰¹¹¹²³,Monti Simona M.¹²³,Supuran Claudiu T.¹⁰¹¹¹²³^ORCID,De Simone Giuseppina¹²³^ORCID

Affiliation:

1. Istituto di Biostrutture e Bioimmagini-CNR

2. Naples

3. Italy

4. Department of Pharmacy

5. “G. d’Annunzio” University of Chieti-Pescara

6. 66100 Chieti

7. Dipartimento di Chimica e Tecnologie del Farmaco

8. Sapienza University of Rome

9. 00185 Rome

10. Neurofarba Department

11. Università degli Studi di Firenze

12. Florence

Abstract

Catechols adopt a peculiar binding mode to the CA active site which involves both the zinc bound water molecule and the “deep water”.

Funder

Regione Campania

Ministero dell’Istruzione, dell’Università e della Ricerca

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2020/CC/D0CC05172A

Reference33 articles.

1. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

2. Carbonic Anhydrase: Zinc and the Mechanism of Catalysis

3. Refined structure of human carbonic anhydrase II at 2.0 Å resolution

4. Interfering with pH regulation in tumours as a therapeutic strategy

5. Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations

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