Potent trifluoromethoxy, trifluoromethylsulfonyl, trifluoromethylthio and pentafluorosulfanyl containing (1,3,4-oxadiazol-2-yl)benzamides against drug-resistant Gram-positive bacteria-Reference-Cited by-同舟云学术

Potent trifluoromethoxy, trifluoromethylsulfonyl, trifluoromethylthio and pentafluorosulfanyl containing (1,3,4-oxadiazol-2-yl)benzamides against drug-resistant Gram-positive bacteria

Published:2020 Issue:1 Volume:11 Page:102-110
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Naclerio George A.¹²³⁴⁵,Abutaleb Nader S.⁶⁷⁴⁵,Onyedibe Kenneth I.¹²³⁴⁵,Seleem Mohamed N.⁶⁷⁴⁵⁸^ORCID,Sintim Herman O.¹²³⁴⁵^ORCID

Affiliation:

1. Department of Chemistry

2. Institute for Drug Discovery

3. Purdue University

4. West Lafayette

5. USA

6. Department of Comparative Pathobiology

7. Purdue University College of Veterinary Medicine

8. Purdue Institute of Inflammation, Immunology, and Infectious Diseases

Abstract

Switching from bacteriostatic against methicillin-resistant S. aureus to bactericidal via SCF₃ or SF₅ substitution.

Funder

Purdue University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/MD/C9MD00391F

Reference43 articles.

1. Staphylococcus aureus Infections: Epidemiology, Pathophysiology, Clinical Manifestations, and Management

2. Waves of resistance: Staphylococcus aureus in the antibiotic era

3. Comparison of Mortality Associated with Methicillin‐Resistant and Methicillin‐SusceptibleStaphylococcus aureusBacteremia: A Meta‐analysis

4. Current Treatment Options for Community‐Acquired Methicillin‐ResistantStaphylococcus aureusInfection

5. Future challenges and treatment of Staphylococcus aureus bacteremia with emphasis on MRSA

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