Phosphate tricyclic coumarin analogs as steroid sulfatase inhibitors: synthesis and biological activity-Reference-Cited by-同舟云学术

Phosphate tricyclic coumarin analogs as steroid sulfatase inhibitors: synthesis and biological activity

Published:2014 Issue:84 Volume:4 Page:44350-44358
ISSN:2046-2069
Container-title:RSC Adv.
language:en
Short-container-title:RSC Adv.

Author:

Kozak Witold¹²³⁴,Daśko Mateusz¹²³⁴,Masłyk Maciej⁵⁶⁷⁸,Pieczykolan Jerzy S.⁹¹⁰¹¹,Gielniewski Bartłomiej⁵⁶⁷⁸,Rachon Janusz¹²³⁴,Demkowicz Sebastian¹²³⁴

Affiliation:

1. Department of Organic Chemistry

2. Chemical Faculty

3. Gdansk University of Technology

4. 80-233 Gdansk, Poland

5. Department of Molecular Biology

6. Faculty of Biotechnology and Environment Sciences

7. The John Paul II Catholic University of Lublin

8. 20-708 Lublin, Poland

9. Drug Discovery Department

10. Adamed Group

11. 05-152 Czosnów, Poland

Abstract

In the present work, we report convenient methods for the synthesis and biological evaluation of phosphate tricyclic coumarin derivatives as potential steroid sulfatase inhibitors.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/RA/C4RA07135B

Reference27 articles.

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3. Steroid sulfatase inhibitors for estrogen- and androgen-dependent cancers

4. Inhibition of Steroid 3-Sulfatase by Endogenous Steroids. A Possible Mechanism Controlling Placental Estrogen Synthesis from Conjugated Precursors1

5. Prognostic significance of aromatase and estrone sulfatase enzymes in human breast cancer

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