Access to acridones by tandem copper(i)-catalyzed electrophilic amination/Ag(i)-mediated oxidative annulation of anthranils with arylboronic acids-Reference-Cited by-同舟云学术

Access to acridones by tandem copper(i)-catalyzed electrophilic amination/Ag(i)-mediated oxidative annulation of anthranils with arylboronic acids

Published:2021 Issue:39 Volume:19 Page:8487-8491
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Jiang Chun-Yong¹²,Xie Hui³,Huang Zhuo-Jun¹,Liang Jing-Yi¹,Huang Yan-Xia¹,Liang Qiu-Ping¹,Zeng Jun-Yi¹,Zhou Binhua²,Zhang Shang-Shi¹³^ORCID,Shu Bing¹

Affiliation:

1. School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou, 510006, P. R. China

2. School of Ethnic Medicine, Guizhou Minzu University, Guiyang, 550025, P. R. China

3. Center for Drug Research and Development, Guangdong Pharmaceutical University, Guangzhou, 510006, P. R. China

Abstract

An efficient and practical approach for the synthesis of medicinally important acridones was developed from anthranils and arylboronic acids by a tandem copper(i)-catalyzed electrophilic amination/Ag(i)-mediated oxidative annulation strategy.

Funder

Guangdong Pharmaceutical University

Natural Science Foundation of Guizhou Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/OB/D1OB01586A

Reference46 articles.

1. Reactivity of the Acridine Ring: A Review

2. Synthesis and Anti-BVDV Activity of Acridones As New Potential Antiviral Agents

3. Antitumor Psoropermum Xanthones and Sarcomelicope Acridones: Privileged Structures Implied in DNA Alkylation

4. Discovery of dual function acridones as a new antimalarial chemotype

5. Recent developments in the synthesis and biological activity of acridine/acridone analogues

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