Straightforward synthesis of enantiomerically pure 1,2,3-triazoles derived from amino esters-Reference-Cited by-同舟云学术

Straightforward synthesis of enantiomerically pure 1,2,3-triazoles derived from amino esters

Published:2018 Issue:17 Volume:16 Page:3168-3176
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Silveira-Dorta Gastón¹²³⁴⁵^ORCID,Jana Sampad¹²³⁴⁵^ORCID,Borkova Lucie⁶⁷⁸⁹¹⁰^ORCID,Thomas Joice¹²³⁴⁵^ORCID,Dehaen Wim¹²³⁴⁵^ORCID

Affiliation:

1. Molecular Design and Synthesis

2. Department of Chemistry

3. KU Leuven

4. B-3001 Leuven

5. Belgium

6. Institute of Molecular and Translational Medicine

7. Faculty of Medicine and Dentistry

8. Palacky University in Olomouc

9. 779 00 Olomouc

10. Czech Republic

Abstract

An easy, good-yielding access to functionalized enantiomerically pure 1,2,3-triazole derivatives of amino acids using commercially available ketones and amino esters is described.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C8OB00533H

Reference27 articles.

1. Synthesis and antiproliferative activity of glutamic acid-based dipeptides

2. Direct Stereoselective Synthesis of Enantiomerically Pure anti-β-Amino Alcohols

3. Synthesis and identification of unprecedented selective inhibitors of CK1ε

4. Design, synthesis, and biological activity of novel triazole amino acids used to probe binding interactions between ligand and neutral amino acid transport protein SN1

5. Click chemistry: function follows form

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