Copper-mediated [3 + 2] oxidative cyclization of oxime acetate and its utility in the formal synthesis of fentiazac-Reference-Cited by-同舟云学术

Copper-mediated [3 + 2] oxidative cyclization of oxime acetate and its utility in the formal synthesis of fentiazac

Published:2024 Issue:3 Volume:22 Page:521-528
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Jadhao Nitin L¹²,Musale Harish B.³,Gajbhiye Jayant M.¹²,Humne Vivek T.³^ORCID

Affiliation:

1. Organic Chemistry Division, CSIR-National Chemical Laboratory, Pune, 411008, India

2. Academy of Scientific and Innovative Research (AcSIR), Ghaziabad, 201002, India

3. Department of Chemistry, Shri R. R. Lahoti Science College, Morshi, 444905, India

Abstract

The direct synthesis of 2-aminothiazole has been developed from oxime acetate using a copper catalyst. The applicability of the present method is used in the formal synthesis of fentiazac.

Funder

CouncilofScientific and Industrial Research, India

Department of Science and Technology, Ministry of Science and Technology

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2024/OB/D3OB01882B

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