A practical synthesis of 2,3-dihydro-1,5-benzothiazepines
Author:
Affiliation:
1. Department of Chemistry
2. Università degli Studi di Milano
3. Milano
4. Italy
5. Department of Pharmaceutical Sciences
Abstract
Hexafluoro-2-propanol as the solvent allows a catalyst free domino approach to 2,3-dihydro-1,5-benzothiazepines in up to 98% yield.
Publisher
Royal Society of Chemistry (RSC)
Subject
Pollution,Environmental Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2017/GC/C7GC02097J
Reference26 articles.
1. 1,5-Benzothiazepine, a versatile pharmacophore: A review
2. 1,5-Benzoheteroazepines through eco-friendly general condensation reactions
3. An Improved Procedure for the Synthesis of 1,5-Benzothiazepines Using Ceric Ammonium Nitrate (CAN)
4. Ga(OTf)3-promoted condensation reactions for 1,5-benzodiazepines and 1,5-benzothiazepines
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