Tuning a modular system – synthesis and characterisation of a boron-rich s-triazine-based carboxylic acid and amine bearing a galactopyranosyl moiety-Reference-Cited by-同舟云学术

Tuning a modular system – synthesis and characterisation of a boron-rich s-triazine-based carboxylic acid and amine bearing a galactopyranosyl moiety

Published:2020 Issue:1 Volume:49 Page:57-69
ISSN:1477-9226
Container-title:Dalton Transactions
language:en
Short-container-title:Dalton Trans.

Author:

Kellert Martin¹²³⁴⁵^ORCID,Hoppenz Paul⁶⁷³⁴⁵^ORCID,Lönnecke Peter¹²³⁴⁵^ORCID,Worm Dennis J.⁶⁷³⁴⁵^ORCID,Riedl Bernd⁸⁹⁵,Koebberling Johannes⁸⁹⁵,Beck-Sickinger Annette G.⁶⁷³⁴⁵^ORCID,Hey-Hawkins Evamarie¹²³⁴⁵^ORCID

Affiliation:

1. Faculty of Chemistry and Mineralogy

2. Institute of Inorganic Chemistry

3. Leipzig University

4. 04103 Leipzig

5. Germany

6. Faculty of Life Sciences

7. Institute of Biochemistry

8. Bayer AG

9. 42113 Wuppertal

Abstract

Introduction of a galactopyranosyl moiety in s-triazine-based boron-rich carboxylic acids and amines results in soluble and suitable coupling partners for tumour-selective biomolecules with applications in boron neutron capture therapy (BNCT).

Funder

European Regional Development Fund

European Commission

Deutsche Forschungsgemeinschaft

Publisher

Royal Society of Chemistry (RSC)

Subject

Inorganic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/DT/C9DT04031E

Reference69 articles.

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