Green synthesis of glutaramides, piperidino[1,2-<i>a</i>]benzimidazol-1-ones and <i>N</i>-cyclopentenyl benzimidazolones enabled by microwave assisted domino reactions of cyclic 2-diazo-1,3-diketones with aniline derivatives-Reference-Cited by-同舟云学术

Green synthesis of glutaramides, piperidino[1,2-a]benzimidazol-1-ones and N-cyclopentenyl benzimidazolones enabled by microwave assisted domino reactions of cyclic 2-diazo-1,3-diketones with aniline derivatives

Published:2024 Issue:16 Volume:11 Page:4516-4521
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Zhao Cheng¹²,Hu Xiao-Wei²,Xu Yi-Bin²,Liu Xiong-Wei¹,Tian You-Ping¹,Liu Yun-Lin²³⁴^ORCID

Affiliation:

1. School of Pharmacy, Guizhou University of Traditional Chinese Medicine, Guiyang 550025, China

2. School of Chemistry and Chemical Engineering, Guangzhou University, 230 Wai Huan Xi Road, Guangzhou, 510006, China

3. Key Laboratory of Tropical Medicinal Resource Chemistry of Ministry of Education; Hainan Normal University, Hainan, Haikou 571158, China

4. Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, School of Chemistry and Molecular Engineering, East China Normal University, 3663 North Zhongshan Rd, Shanghai, 200062, China

Abstract

Microwave-assisted divergent domino reactions between cyclic 2-diazo-1,3-diketones and aniline derivatives selectively leading to either glutaramides, piperidino[1,2-a]benzimidazol-1-ones or N-cyclopentenyl benzimidazolones are developed.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Guangdong Province

National College Students Innovation and Entrepreneurship Training Program

Hainan Normal University

East China Normal University

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/QO/D4QO00613E

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