Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: synthesis and antimycobacterial evaluation-Reference-Cited by-同舟云学术

Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: synthesis and antimycobacterial evaluation

Published:2015 Issue:7 Volume:6 Page:1311-1317
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Servusova-Vanaskova Barbora¹²³⁴⁵,Jandourek Ondrej¹²³⁴⁵,Paterova Pavla¹²³⁴⁵,Kordulakova Jana⁶⁷⁸⁹,Plevakova Magdalena¹²³⁴⁵,Kubicek Vladimir¹²³⁴⁵,Kucera Radim¹²³⁴⁵,Garaj Vladimir¹⁰⁷¹¹⁹,Naesens Lieve¹²¹³¹⁴¹⁵,Kunes Jiri¹²³⁴⁵,Dolezal Martin¹²³⁴⁵,Zitko Jan¹²³⁴⁵

Affiliation:

1. Faculty of Pharmacy in Hradec Králové

2. Charles University in Prague

3. Heyrovského 1203

4. Hradec Králové 500 05

5. Czech Republic

6. Faculty of Natural Sciences

7. Comenius University

8. 842 15 Bratislava

9. Slovakia

10. Faculty of Pharmacy

11. Bratislava

12. Rega Institute for Medical Research

13. KU Leuven

14. Leuven

15. Belgium

Abstract

A series of alkylamino derivatives ofN-benzylpyrazine-2-carboxamide was designed, synthesized and assayedin vitrofor their antimycobacterial activity.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/MD/C5MD00178A

Reference31 articles.

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2. World Health Organization , Global Tuberculosis, Report 2012. WHO/HTM/TB/2012.6

3. World Health Organization , Global Tuberculosis, Report 2014. WHO/HTM/TB/2014.08

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