Practical synthesis and biological screening of sulfonyl hydrazides-Reference-Cited by-同舟云学术

Practical synthesis and biological screening of sulfonyl hydrazides

Published:2023 Issue:10 Volume:21 Page:2118-2126
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Macara João¹,Caldeira Catarina¹,Cunha José¹^ORCID,Coelho Jaime A. S.²^ORCID,Silva Maria J. S. A.³^ORCID,Krämer Konrad⁴⁵,Grathwol Christoph W.⁴⁵,Bräse Stefan⁴⁵,Marques M. Manuel B.¹^ORCID

Affiliation:

1. LAQV@REQUIMTE, Departamento de Química, NOVA School of Science and Technology, Universidade Nova de Lisboa, Campus de Caparica, 2829-516 Caparica, Portugal

2. Centro de Química Estrutural, Faculdade de Ciências, Universidade de Lisboa, Campo Grande, Lisboa 1749-016, Portugal

3. Research Institute for Medicines (iMed.ULisboa), Faculty of Pharmacy, Universidade de Lisboa, Av. Prof. Gama Pinto, 1649-003, Lisboa, Portugal

4. Institute of Organic Chemistry, Organic Chemistry I, Fritz-Haber-Weg 6, 76131 Karlsruhe, Germany

5. Institute of Biological and Chemical Systems – Functional Molecular Systems (IBCS-FMS), Hermann-von-Helmholtz-Platz 1, D-76344 Eggenstein-Leopoldshafen, Germany

Abstract

A hypervalent iodine-mediated synthesis of sulfonyl hydrazides is described. The methodology relies on the umpolung reactivity of benziodoxolone reagents. Mechanistic studies and biological screening were performed.

Funder

Fundação para a Ciência e a Tecnologia

Laboratório Associado para a Química Verde

European Regional Development Fund

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/OB/D2OB02160A

Reference27 articles.

1. Sulfonyl Hydrazides in Organic Synthesis: A Review of Recent Studies

2. Hydroxysulfonylation of alkenes: an update

3. Nine-step total synthesis of (−)-strychnofoline

4. Sulfonyl hydrazides as sulfonyl sources in organic synthesis

5. Novel 10-I-3 Hypervalent Iodine-Based Compounds for Electrophilic Trifluoromethylation

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Visible‐Light‐Driven Sulfonamidation of Arylazo Sulfonesthrough One‐Pot Multicomponent Reaction;Asian Journal of Organic Chemistry;2023-07-24