A novel series of dipeptide derivatives containing indole-3-carboxylic acid conjugates as potential antimicrobial agents: the design, solid phase peptide synthesis, <i>in vitro</i> biological evaluation, and molecular docking study-Reference-Cited by-同舟云学术

A novel series of dipeptide derivatives containing indole-3-carboxylic acid conjugates as potential antimicrobial agents: the design, solid phase peptide synthesis, in vitro biological evaluation, and molecular docking study

Published:2023 Issue:35 Volume:13 Page:24250-24263
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Tivari Sunil R.¹,Kokate Siddhant V.²,Delgado-Alvarado Enrique³⁴,Gayke Manoj S.⁵,Kotmale Amol⁶,Patel Harun⁷,Ahmad Iqrar⁷,Sobhia Elizabeth M.⁸,Kumar Siva G.⁹,Lara Bianey García²,Jain Vicky D.¹,Jadeja Yashwantsinh¹^ORCID

Affiliation:

1. Department of Chemistry, Marwadi University, Rajkot-360003, Gujarat, India

2. Departamento de Química, Universidad de Guanajuato, Noria Alta S/N, Guanajuato-36050, Guanajuato, Mexico

3. Micro and Nanotechnology Research Center, Universidad Veracruzana, Blvd. Av. Ruiz Cortines No. 455 Fracc. Costa Verde, Boca del Río 94294, Mexico

4. Facultad de Ciencias Quimicas, Universidad Veracruzana, Blvd. Av. Ruiz Cortines No. 455 Fracc. Costa Verde, Boca del Río 94294, Mexico

5. Indrashil University, Rajpur, Kadi, Mehsana 382740, Gujarat, India

6. Department of Chemistry, Savitribai Phule Pune University, Pune 411007, Maharashtra, India

7. Department of Pharmaceutical Chemistry, R C. Patel Institute of Pharmaceutical Education and Research, Shirpur District, Dhule 425405, Maharashtra, India

8. Department of Pharmacoinformatics, NIPER, Mohali 160062, Punjab, India

9. Department of Medicinal Chemistry, Sri Venkateswara College of Pharmacy, Chittoor 517127, Andhra Pradesh, India

Abstract

A new library of peptide-heterocycle hybrids consisting of an indole-3-carboxylic acid constituent conjugated with short dipeptide motifs was designed and synthesized by using the solid phase peptide synthesis methodology.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/RA/D3RA04100J

Reference71 articles.

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3. J.O'Neill , Tackling drug-resistant infections globally: final report and recommendations , Review on Antimicrobial Resistance , London , 2016

4. WHO , Antimicrobial resistance , accessed Jan 08, 2023, 2021 , https://www.who.int/newsroom/factsheets/detail/antimicrobial-resistance

5. Antimicrobial resistance: a global multifaceted phenomenon

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