Regioselective N-1 and C-2 diacylation of 3-substituted indoles with arylglyoxal hydrates for the synthesis of indolyl diketones-Reference-Cited by-同舟云学术

Regioselective N-1 and C-2 diacylation of 3-substituted indoles with arylglyoxal hydrates for the synthesis of indolyl diketones

Published:2018 Issue:38 Volume:16 Page:6998-7003
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Pan Dalong¹²³⁴⁵,Chu Jinpeng¹²³⁴⁵,Gao Xianrui¹²³⁴⁵,Wang Cuiping¹²³⁴⁵^ORCID,Meng Qingtao¹²³⁴⁵^ORCID,Chi Haijun¹²³⁴⁵,Dong Yan¹²³⁴⁵,Duan Chunying⁶⁷⁸⁵^ORCID,Zhang Zhiqiang¹²³⁴⁵^ORCID

Affiliation:

1. Key Laboratory for Functional Material

2. Educational Department of Liaoning Province

3. University of Science and Technology Liaoning

4. Anshan 114051

5. P. R. China

6. State Key Laboratory of Fine Chemicals

7. Dalian University of Technology

8. Dalian

Abstract

A highly regioselective N-1 and C-2 diacylation of 3-substituted indoles with arylglyoxal hydrates to afford N-1 and C-2 indolyl diketones in moderate to good yields is described.

Funder

National Natural Science Foundation of China

Department of Education of Liaoning Province

University of Science and Technology Liaoning

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C8OB01776J

Reference59 articles.

1. R. J. Sundberg , Indoles , Academic Press , London, UK , 1996