6-Deoxy-6-fluoro galactofuranosides: regioselective glycosylation, unexpected reactivity, and anti-leishmanial activity-Reference-Cited by-同舟云学术

6-Deoxy-6-fluoro galactofuranosides: regioselective glycosylation, unexpected reactivity, and anti-leishmanial activity

Published:2020 Issue:7 Volume:18 Page:1462-1475
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Vaugenot Jeane¹²³⁴⁵,El Harras Abderrafek¹²³⁴⁵,Tasseau Olivier¹²³⁴⁵,Marchal Rémi¹²³⁴⁵,Legentil Laurent¹²³⁴⁵^ORCID,Le Guennic Boris¹²³⁴⁵^ORCID,Benvegnu Thierry¹²³⁴⁵,Ferrières Vincent¹²³⁴⁵^ORCID

Affiliation:

1. Univ Rennes

2. Ecole Nationale Supérieure de Chimie de Rennes

3. CNRS

4. F-35000 Rennes

5. France

Abstract

Standard glycosylation of unprotected 6-fluorogalactofuranoside turned to three competitive reactions and afforded difuranosides able to impact growth of Leishmania tarentolae.

Funder

Centre National de la Recherche Scientifique

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/C9OB02596K

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