HFIP-promoted Michael reactions: direct para-selective C–H activation of anilines with maleimides-Reference-Cited by-同舟云学术

HFIP-promoted Michael reactions: direct para-selective C–H activation of anilines with maleimides

Published:2019 Issue:8 Volume:17 Page:2242-2246
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Li Bang¹²³⁴⁵,Mao Qi¹²³⁴⁵,Zhou Jia⁶⁷⁸⁹¹⁰,Liu Feng¹²³⁴⁵^ORCID,Ye Na¹²³⁴⁵^ORCID

Affiliation:

1. Department of Medicinal Chemistry

2. Jiangsu Key Laboratory of Neuropsychiatric Diseases and College of Pharmaceutical Sciences

3. Soochow University

4. Suzhou

5. People's Republic of China

6. Department of Pharmacology and Toxicology

7. Center for Addiction Research

8. University of Texas Medical Branch

9. Galveston

10. USA

Abstract

Diversified 3-aryl succinimide derivatives are efficiently and selectively prepared from various N,N-disubstituted anilines and maleimides under facile metal-free conditions.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Jiangsu Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C8OB03073A

Reference62 articles.

1. Rapid Evaluation ofAntrodia camphorataNatural Products and Derivatives in Tumourigenic Liver Progenitor Cells with a Novel Cell Proliferation Assay

2. Microwave-assisted synthesis and biological evaluation of 3,4-diaryl maleic anhydride/N-substituted maleimide derivatives as combretastatin A-4 analogues

3. Ruthenium(II)-Catalyzed Hydroarylation of Maleimides Using Carboxylic Acids as a Traceless Directing Group

4. An Optimized RAD51 Inhibitor That Disrupts Homologous Recombination without Requiring Michael Acceptor Reactivity

5. Synthesis and anticancer activity of nitrosourea derivatives of phensuximide

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