One step stereoselective synthesis of oxazoline-fused saccharides and their conversion into the corresponding 1,2-cis glycosylamines bearing various protected groups-Reference-Cited by-同舟云学术

One step stereoselective synthesis of oxazoline-fused saccharides and their conversion into the corresponding 1,2-cis glycosylamines bearing various protected groups

Published:2021 Issue:7 Volume:19 Page:1580-1588
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Dong Sanfeng¹²³⁴⁵,Zhao Yitian¹²³⁴⁵,Shi Yulong⁴⁵⁶²³,Xu Zhijian⁴⁵⁶²³^ORCID,Shen Jingshan⁴⁵⁶²³^ORCID,Jia Qi¹²³,Li Yiming¹²³,Chen Kaixian¹²³⁴⁵,Li Bo⁴⁵⁶²³^ORCID,Zhu Weiliang¹²³⁴⁵^ORCID

Affiliation:

1. Shanghai University of Traditional Chinese Medicine

2. Shanghai 201203

3. China

4. CAS Key Laboratory of Receptor Research; Drug Discovery and Design Center

5. Shanghai Institute of Materia Medica

6. Chinese Academy of Sciences

Abstract

Oxazolinoses, which can be converted into 1,2-cis glycosylamines and allowed the access to schisandrin derivatives, are prepared concisely from peracetylated saccharides and benzonitriles under acidic conditions with stoichiometric amounts of water.

Funder

National Natural Science Foundation of China

National Science and Technology Major Project

Natural Science Foundation of Shanghai

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/OB/D0OB02477E

Reference33 articles.

1. Glycans in drug discovery