Synthesis of tri(di)fluoroethylanilines via copper-catalyzed coupling reaction of tri(di)fluoroethylamine with (hetero)aromatic bromides-Reference-Cited by-同舟云学术

Synthesis of tri(di)fluoroethylanilines via copper-catalyzed coupling reaction of tri(di)fluoroethylamine with (hetero)aromatic bromides

Published:2019 Issue:45 Volume:17 Page:9799-9807
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Chen Suo¹²³⁴⁵,Wang Hui¹²³⁴⁵,Jiang Wei⁶⁷⁴,Rui Pei-Xin¹²³⁴,Hu Xiang-Guo¹²³⁴⁵^ORCID

Affiliation:

1. National Engineering Research Center for Carbohydrate Synthesis

2. Jiangxi Normal University

3. Nanchang

4. China

5. Key Laboratory of Small Functional Organic Molecule

6. Research Center for Traditional Chinese Medicine Resources and Ethnic Minority Medicine

7. Jiangxi University of Traditional Chinese Medicine

Abstract

A practical and efficient synthesis of fluoroalkylanilines has been achieved via the Ullmann type coupling of (hetero)aromatic bromides with tri(di)fluoroethylamine.

Funder

Natural Science Foundation of Jiangxi Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C9OB02271F

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