Uncatalysed diaryldiazo cyclopropanations on bicyclic lactams: access to annulated prolines-Reference-Cited by-同舟云学术

Uncatalysed diaryldiazo cyclopropanations on bicyclic lactams: access to annulated prolines

Published:2015 Issue:23 Volume:13 Page:6522-6550
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Harris Lawrence¹²³⁴⁵,Gilpin Martin⁶⁷⁵,Thompson Amber L.¹²³⁴⁵,Cowley Andrew R.¹²³⁴⁵,Moloney Mark G.¹²³⁴⁵

Affiliation:

1. The Department of Chemistry

2. Chemistry Research Laboratory

3. The University of Oxford

4. Oxford

5. UK

6. GlaxoSmithKline Research & Development Ltd

7. Harlow

Abstract

The uncatalysed cycloaddition of substituted diaryldiazo compounds onto bicyclic unsaturated lactams derived from pyroglutamic acid efficiently leads to highly functionalised azatricyclononanes.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00648A

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