Diastereoselective approach to rationally design tetrahydro-β-carboline–isatin conjugates as potential SERMs against breast cancer-Reference-Cited by-同舟云学术

Diastereoselective approach to rationally design tetrahydro-β-carboline–isatin conjugates as potential SERMs against breast cancer

Published:2019 Issue:17 Volume:9 Page:9809-9819
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Sharma Bharvi¹²³⁴,Singh Amandeep¹²³⁴,Gu Liang⁵⁶⁷⁸,Saha Sourav Taru⁵⁶⁷⁸,Singh-Pillay Ashona⁹¹⁰¹¹⁸,Cele Nosipho⁹¹⁰¹¹⁸,Singh Parvesh⁹¹⁰¹¹⁸,Kaur Mandeep⁵⁶⁷⁸,Kumar Vipan¹²³⁴^ORCID

Affiliation:

1. Department of Chemistry

2. Guru Nanak Dev University

3. Amritsar-143005

4. India

5. School of Molecular and Cell Biology

6. University of the Witwatersrand

7. Johannesburg

8. South Africa

9. School of Chemistry and Physics

10. University of KwaZulu Natal

11. Durban 4000

Abstract

A series of tetrahydro-β-carboline–isatin conjugates was prepared and assayed for anti-proliferative activities on Estrogen Responsive ER(+) and non-responsive ER(−ve) cell-lines.

Funder

Council for Scientific and Industrial Research

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/RA/C9RA00744J

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