Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines to develop functionalized ligands to target adenosine receptors: fluorescent ligands as an example-Reference-Cited by-同舟云学术

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Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines to develop functionalized ligands to target adenosine receptors: fluorescent ligands as an example

Published:2019 Issue:7 Volume:10 Page:1094-1108
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Federico Stephanie¹²³⁴^ORCID,Margiotta Enrico⁵⁶⁷⁸⁴,Paoletta Silvia⁵⁶⁷⁸⁴,Kachler Sonja⁹¹⁰¹¹¹²,Klotz Karl-Norbert⁹¹⁰¹¹¹²^ORCID,Jacobson Kenneth A.¹³¹⁴¹⁵¹⁶¹⁷^ORCID,Pastorin Giorgia¹⁸¹⁹²⁰^ORCID,Moro Stefano⁵⁶⁷⁸⁴^ORCID,Spalluto Giampiero¹²³⁴^ORCID

Affiliation:

1. Department of Chemical and Pharmaceutical Sciences

2. University of Trieste

3. 34127 Trieste

4. Italy

5. Molecular Modeling Section (MMS)

6. Dipartimento di Scienze del Farmaco

7. Università degli Studi di Padova

8. 35131 Padova

9. Institut für Pharmakologie und Toxicologie

10. Universität Würzburg

11. 97078 Würzburg

12. Germany

13. Laboratory of Bioorganic Chemistry

14. National Institute of Diabetes and Digestive and Kidney Diseases

15. National Institutes of Health

16. Bethesda

17. USA

18. Department of Pharmacy

19. National University of Singapore

20. 117543 Singapore

Abstract

A series of adenosine receptor antagonists bearing a reactive linker was developed.

Funder

National Institute of Diabetes and Digestive and Kidney Diseases

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/MD/C9MD00014C

Reference51 articles.

1. Probing the pharmacology of G protein-coupled receptors with fluorescent ligands

2. Emerging concepts in molecular MRI

3. Ligand conjugation: An emerging platform for enhanced brain drug delivery

4. Ligand-Targeted Drug Delivery

5. Polymer Therapeutics: Concepts and Applications

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3. Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine A₃ Receptor Expression;Journal of Medicinal Chemistry;2023-08-02

4. One-pot synthesis of novel pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines under microwave irradiation in a green solvent;Tetrahedron;2023-07

5. Adenosine Receptor Ligands, Probes, and Functional Conjugates: A 20-Year History of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidines (PTP);Topics in Medicinal Chemistry;2023

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