A structure guided drug-discovery approach towards identification of Plasmodium inhibitors
Author:
Affiliation:
1. Medicinal Chemistry Lab
2. Department of Biosciences
3. Jamia Millia Islamia (A Central University)
4. New Delhi 110025
5. India
6. Protein Conformation and Enzymology Lab
Abstract
This article provides a comprehensive review of inhibitors from natural, semisynthetic or synthetic sources against key targets ofPlasmodium falciparum.
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/RA/C5RA19673F
Reference212 articles.
1. Synthesis and biological evaluation of some novel pyrido[1,2-a]pyrimidin-4-ones as antimalarial agents
2. WHO Report, 2014. http://apps.who.int/iris/bitstream/10665/144852/2/9789241564830_eng.pdf
3. Plasmodium falciparum Plasmepsin V ( Pf PMV): Insights into recombinant expression, substrate specificity and active site structure
4. Metalloantimalarials
5. Antimalarial drug discovery: efficacy models for compound screening
Cited by 21 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Diversified Synthesis of N-Benzoyl Piperidine Tetraoxane Analogues Using Molybdenum Trioxide as a Newer Catalyst and Its Antiplasmodial Activity;ACS Omega;2024-07-12
2. Redox modulating small molecules having antimalarial efficacy;Biochemical Pharmacology;2023-12
3. New structural classes of antimalarials;European Journal of Medicinal Chemistry;2022-11
4. Target-Based Virtual Screening of Natural Compounds Identifies a Potent Antimalarial With Selective Falcipain-2 Inhibitory Activity;Frontiers in Pharmacology;2022-04-06
5. Structure- and ligand-based drug design methods for the modeling of antimalarial agents: a review of updates from 2012 onwards;Journal of Biomolecular Structure and Dynamics;2021-06-15
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3