An Ullmann N-arylation/2-amidation cascade by self-relay copper catalysis: one-pot synthesis of indolo[1,2-a]quinazolinones-Reference-Cited by-同舟云学术

An Ullmann N-arylation/2-amidation cascade by self-relay copper catalysis: one-pot synthesis of indolo[1,2-a]quinazolinones

Published:2017 Issue:11 Volume:4 Page:2124-2127
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Abe Takumi¹²³⁴^ORCID,Takahashi Yuka¹²³⁴,Matsubara Yuki¹²³⁴,Yamada Koji¹²³⁴

Affiliation:

1. Faculty of Pharmaceutical Sciences

2. Health Sciences University of Hokkaido

3. Ishikari-tobetsu

4. Japan

Abstract

We have developed a self-relay copper(i)-catalyzed Ullmann N-arylation/2-amidation cascade to form functionalized indolo[1,2-a]quinazolinones in one-pot from easily available indoles with 2-bromobenzamides.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/QO/C7QO00549K

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