Stereoselective, solvent free, highly efficient synthesis of aldo- and keto-N-acylhydrazones applying grindstone chemistry-Reference-Cited by-同舟云学术

Stereoselective, solvent free, highly efficient synthesis of aldo- and keto-N-acylhydrazones applying grindstone chemistry

Published:2017 Issue:9 Volume:19 Page:2212-2224
ISSN:1463-9262
Container-title:Green Chemistry
language:en
Short-container-title:Green Chem.

Author:

dos Santos Filho José Maurício¹²³⁴⁵^ORCID,Pinheiro Savio Moita⁶⁷⁸⁹⁵

Affiliation:

1. Laboratory of Design and Synthesis Applied to Medicinal Chemistry-SintMed®

2. Centro de Tecnologia e Geociências

3. Universidade Federal de Pernambuco

4. Recife

5. Brazil

6. Departamento de Química

7. Centro de Ciências Exatas e da Natureza

8. Universidade Federal da Paraíba

9. João Pessoa

Abstract

An efficient and stereoselective methodology for the synthesis of N-acylhydrazones is disclosed, based on grindstone chemistry. The method tolerates a broad variety of substrates, as demonstrated by the 51 examples, 21 of them unpublished.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pollution,Environmental Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/GC/C7GC00730B

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