Convergent synthesis, kinetics insight and allosteric computational ascriptions of thiazole-(5-aryl)oxadiazole hybrids embraced with propanamides as alkaline phosphatase inhibitors-Reference-Cited by-同舟云学术

Convergent synthesis, kinetics insight and allosteric computational ascriptions of thiazole-(5-aryl)oxadiazole hybrids embraced with propanamides as alkaline phosphatase inhibitors

Published:2023 Issue:20 Volume:13 Page:13798-13808
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Butt Abdul Rehman Sadiq¹,Abbasi Muhammad Athar¹^ORCID,Aziz-ur-Rehman ¹,Siddiqui Sabahat Zahra¹,Muhammad Shabbir²^ORCID,Raza Hussain³^ORCID,Shah Syed Adnan Ali⁴⁵,Shahid Muhammad⁶,Alsehemi Abdullah G.²^ORCID,Kim Song Ja³^ORCID

Affiliation:

1. Department of Chemistry, Government College University, Lahore 54000, Pakistan

2. Department of Chemistry, College of Science, King Khalid University, P.O. Box 9004, Abha 61413, Saudi Arabia

3. College of Natural Sciences, Department of Biological Sciences, Kongju National University, Gongju, 32588, South Korea

4. Faculty of Pharmacy, Universiti Teknologi MARA Cawangan Selangor Kampus Puncak Alam, Bandar Puncak Alam 42300, Selangor, Malaysia

5. Atta-ur-Rahman Institute for Natural Product Discovery (AuRIns), Universiti Teknologi MARA Cawangan Selangor Kampus Puncak Alam, Bandar Puncak Alam 42300, Selangor, Malaysia

6. Department of Biochemistry, University of Agriculture, Faisalabad 38040, Pakistan

Abstract

Considering the varied pharmacological prominence of thiazole and oxadiazole heterocyclic moieties, a unique series of bi-heterocyclic hybrids, 8a–h, was synthesized in a convergent manner.

Funder

National Research Foundation of Korea

King Khalid University

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/RA/D3RA01348K

Reference42 articles.

1. Novel 1,2,4-triazole analogues as mushroom tyrosinase inhibitors: synthesis, kinetic mechanism, cytotoxicity and computational studies

2. Recent developments of 2-aminothiazoles in medicinal chemistry

3. Efficient Synthesis of 2-Aminothiazoles and Fanetizole in Liquid PEG-400 at Ambient Conditions

4. Synthetic Utility of Ethylidenethiosemicarbazide: Synthesis and Anticancer Activity of 1,3-Thiazines and Thiazoles with Imidazole Moiety

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