Novel cocrystals of the potent 1,2,4-thiadiazole-based neuroprotector with carboxylic acids: virtual screening, crystal structures and solubility performance-Reference-Cited by-同舟云学术

Novel cocrystals of the potent 1,2,4-thiadiazole-based neuroprotector with carboxylic acids: virtual screening, crystal structures and solubility performance

Published:2021 Issue:6 Volume:45 Page:3034-3047
ISSN:1144-0546
Container-title:New Journal of Chemistry
language:en
Short-container-title:New J. Chem.

Author:

Surov Artem O.¹²³^ORCID,Voronin Alexander P.¹²³^ORCID,Vasilev Nikita A.¹²³^ORCID,Ilyukhin Andrey B.⁴⁵³^ORCID,Perlovich German L.¹²³^ORCID

Affiliation:

1. G. A. Krestov Institute of Solution Chemistry of the Russian Academy of Sciences

2. 153045 Ivanovo

3. Russia

4. Institute of General and Inorganic Chemistry RAS

5. Moscow

Abstract

Five new multicomponent solid forms of the biologically active 1,2,4-thiadiazole derivative (TDZH) with dicarboxylic and hydroxybenzoic acids have been discovered by combined virtual/experimental cocrystal screening.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,General Chemistry,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2021/NJ/D0NJ05644H

Reference77 articles.

1. Pharmaceutical cocrystals: from serendipity to design to application

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5. Cocrystals to facilitate delivery of poorly soluble compounds beyond-rule-of-5

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