Binding-induced, turn-on fluorescence of the EGFR/ERBB kinase inhibitor, lapatinib
Author:
Affiliation:
1. Department of Chemistry
2. University of Miami
3. Coral Gables
4. USA
5. Department of Biochemistry and Molecular Biology
6. Miami
Abstract
The photophysical properties, fluorescence imaging, cellular uptake and distribution of lapatinib, an EGFR/ERBB inhibitor are reported.
Funder
National Cancer Institute
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00239G
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