Facile synthesis of 1,4-benzodiazepine-2,5-diones and quinazolinones from amino acids as anti-tubercular agents
Author:
Affiliation:
1. Department of Studies in Chemistry
2. University of Mysore
3. Manasagangothri
4. Mysuru
5. India
6. Adichunchanagiri Institute for Molecular Medicine
7. Nagamangala
8. Department of Studies in Organic chemistry
9. Sri Ram Chem
Abstract
A family of 1,4-benzodiazepine-2,5-diones and quinazolinones with diverse substituents at C-3 position are synthesized by novel, simple and convenient methodology using H2PtCl6as catalyst and were all screened for anti-TB activity.
Funder
University Grants Commission
Publisher
Royal Society of Chemistry (RSC)
Subject
Materials Chemistry,General Chemistry,Catalysis
Link
http://pubs.rsc.org/en/content/articlepdf/2019/NJ/C8NJ04936J
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4. On-Line Synthesis of Pseudopeptide Library Incorporating a Benzodiazepinone Turn Mimic: Biological Evaluation on MC1 Receptors
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