Synthesis of functionalised azepanes and piperidines from bicyclic halogenated aminocyclopropane derivatives-Reference-Cited by-同舟云学术

Synthesis of functionalised azepanes and piperidines from bicyclic halogenated aminocyclopropane derivatives

Published:2017 Issue:25 Volume:15 Page:5364-5372
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Chen Cheng¹²³⁴⁵,Kattanguru Pullaiah¹²³⁴⁵,Tomashenko Olesya A.¹²³⁴⁵,Karpowicz Rafał¹²³⁴⁵,Siemiaszko Gabriela¹²³⁴⁵,Bhattacharya Ahanjit¹²³⁴⁵,Calasans Vinícius¹²³⁴⁵,Six Yvan¹²³⁴⁵^ORCID

Affiliation:

1. Laboratoire de Synthèse Organique (LSO)

2. UMR 7652 CNRS/ENSTA/École Polytechnique

3. Université Paris-Saclay

4. 91128 Palaiseau Cedex

5. France

Abstract

Reductive amination of aldehydes or ketones with suitable dihalogenated bicyclic aminocyclopropanes gives functionalised ring-expanded products in a single step.

Funder

Agence Nationale de la Recherche

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/OB/C7OB01238A

Reference57 articles.

1. The Formal [3+2+1] Cyclisation of Cyclopropylamines with Carboxylic Anhydrides: A Quick Access to Polysubstituted 2,3,3a,4-Tetrahydro6(5H)-indolone Ring Systems

2. The Intramolecular Aromatic Electrophilic Substitution of Aminocyclopropanes Prepared by the Kulinkovich-de Meijere Reaction

3. Aminocyclopropanes as precursors of endoperoxides with antimalarial activity