Sulfonyl radical-enabled 6-endo-trig cyclization for regiospecific synthesis of unsymmetrical diaryl sulfones-Reference-Cited by-同舟云学术

Sulfonyl radical-enabled 6-endo-trig cyclization for regiospecific synthesis of unsymmetrical diaryl sulfones

Published:2016 Issue:11 Volume:3 Page:1452-1456
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Fu Rong¹²³⁴⁵,Hao Wen-Juan¹²³⁴⁵,Wu Ya-Nan¹²³⁴⁵,Wang Nan-Nan¹²³⁴⁵,Tu Shu-Jiang¹²³⁴⁵,Li Guigen⁶⁷⁸⁹¹⁰,Jiang Bo¹²³⁴⁵^ORCID

Affiliation:

1. School of Chemistry and Chemical Engineering

2. Jiangsu Key Laboratory of Green Synthetic Chemistry for Functional Materials

3. Jiangsu Normal University

4. Xuzhou 221116

5. P. R. China

6. Department of Chemistry and Biochemistry

7. Texas Tech University

8. Lubbock

9. USA

10. Institute of Chemistry & BioMedical Sciences

Abstract

A new sulfonyl radical-triggered 6-endo-trig cyclization of unactivated 1,5-enynes under catalytic oxidation conditions for flexible synthesis of unprecedented unsymmetrical diaryl sulfones was established.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/QO/C6QO00422A

Reference60 articles.

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3. 5-Chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase

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5. THE REACTION BETWEEN ARYL SULFONATES AND ORGANOMAGNESIUM HALIDES

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