A biocompatible stapling reaction for in situ generation of constrained peptides-Reference-Cited by-同舟云学术

A biocompatible stapling reaction for in situ generation of constrained peptides

Published:2021 Issue:2 Volume:12 Page:669-674
ISSN:2041-6520
Container-title:Chemical Science
language:en
Short-container-title:Chem. Sci.

Author:

Morewood Richard¹²³⁴^ORCID,Nitsche Christoph¹²³⁴^ORCID

Affiliation:

1. Research School of Chemistry

2. Australian National University

3. Canberra

4. Australia

Abstract

A synthetically straightforward and biocompatible peptide-stapling strategy that can be used directly in biochemical assays to identify constrained enzyme inhibitors.

Funder

Australian Research Council

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/SC/D0SC05125J

Reference30 articles.

1. Constrained peptides' time to shine?

2. Constrained Peptides in Drug Discovery and Development

3. Peptide stapling techniques based on different macrocyclisation chemistries

4. Stapled Helical Peptides Bearing Different Anchoring Residues

5. Two-Component Stapling of Biologically Active and Conformationally Constrained Peptides: Past, Present, and Future

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