Evaluation of A-ring fused pyridine d-modified androstane derivatives for antiproliferative and aldo–keto reductase 1C3 inhibitory activity-Reference-Cited by-同舟云学术

Evaluation of A-ring fused pyridine d-modified androstane derivatives for antiproliferative and aldo–keto reductase 1C3 inhibitory activity

Published:2018 Issue:6 Volume:9 Page:969-981
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Savić Marina P.¹²³⁴⁵^ORCID,Ajduković Jovana J.¹²³⁴⁵^ORCID,Plavša Jovana J.⁶²³⁴⁵,Bekić Sofija S.¹²³⁴⁵,Ćelić Andjelka S.⁶²³⁴⁵,Klisurić Olivera R.⁷²³⁴⁵,Jakimov Dimitar S.⁸⁹³¹⁰⁵,Petri Edward T.⁶²³⁴⁵^ORCID,Djurendić Evgenija A.¹²³⁴⁵

Affiliation:

1. Department of Chemistry, Biochemistry and Environmental Protection

2. Faculty of Sciences

3. University of Novi Sad

4. 21000 Novi Sad

5. Serbia

6. Department of Biology and Ecology

7. Department of Physics

8. Oncology Institute of Vojvodina

9. Faculty of Medicine

10. 21204 Sremska Kamenica

Abstract

New A-ring pyridine fused androstanes in d-homo lactone, 17α-picolyl or 17(E)-picolinylidene series were synthesized and validated.

Funder

Ministarstvo Prosvete, Nauke i Tehnološkog Razvoja

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/MD/C8MD00077H

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