Unveiling epidithiodiketopiperazine as a non-histone arginine methyltransferase inhibitor by chemical protein methylome analyses-Reference-Cited by-同舟云学术

Unveiling epidithiodiketopiperazine as a non-histone arginine methyltransferase inhibitor by chemical protein methylome analyses

Published:2018 Issue:66 Volume:54 Page:9202-9205
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Sohtome Yoshihiro¹²³⁴⁵^ORCID,Shimazu Tadahiro⁶²⁴,Barjau Joaquin¹²³⁴,Fujishiro Shinya¹²³⁴,Akakabe Mai¹²³⁴,Terayama Naoki¹²³⁴⁵,Dodo Kosuke¹²³⁴⁵^ORCID,Ito Akihiro⁵⁴⁷⁸⁴,Yoshida Minoru⁵⁴⁹¹⁰¹¹,Shinkai Yoichi⁶²⁴,Sodeoka Mikiko¹²³⁴⁵^ORCID

Affiliation:

1. Synthetic Organic Chemistry Laboratory

2. RIKEN Cluster for Pioneering Research

3. Saitama 351-0198

4. Japan

5. RIKEN Center for Sustainable Resource Science, RIKEN

6. Cellular Memory Laboratory

7. School of Life Sciences

8. Tokyo University of Pharmacy and Life Sciences

9. Department of Biotechnology

10. Graduate School of Agricultural Life Sciences

11. The University of Tokyo

Abstract

We present a chemical methylome analysis to evaluate the inhibitory activity of small molecules towards poorly characterized protein methyltransferases.

Funder

RIKEN

Japan Agency for Medical Research and Development

Japan Society for the Promotion of Science

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2018/CC/C8CC03907K

Reference53 articles.

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2. Selective Inhibitors of Protein Methyltransferases

3. Chemical Probes of Histone Lysine Methyltransferases

4. Mind the Methyl: Methyllysine Binding Proteins in Epigenetic Regulation

5. Histone methylation: a dynamic mark in health, disease and inheritance

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