An efficient approach to 4-chloro quinolines via TMSCl-mediated cascade cyclization of ortho-propynol phenyl azides-Reference-Cited by-同舟云学术

An efficient approach to 4-chloro quinolines via TMSCl-mediated cascade cyclization of ortho-propynol phenyl azides

Published:2018 Issue:9 Volume:5 Page:1537-1541
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Song Xian-Rong¹²³⁴⁵^ORCID,Li Ren¹²³⁴⁵,Ding Haixin¹²³⁴⁵,Chen Xi¹²³⁴⁵,Yang Tao¹²³⁴⁵,Bai Jiang¹²³⁴⁵,Xiao Qiang¹²³⁴⁵^ORCID,Liang Yong-Min⁶⁷⁸⁵^ORCID

Affiliation:

1. Institute of Organic Chemistry

2. Jiangxi Science & Technology Normal University

3. Key Laboratory of Organic Chemistry

4. Nanchang 330013

5. China

6. State Key Laboratory of Applied Organic Chemistry

7. Lanzhou University

8. Lanzhou 730000

Abstract

A novel and efficient strategy for the synthesis of 4-chloro quinolines via the TMSCl-mediated cascade cyclization of easily prepared ortho-propynol phenyl azides is developed.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Jiangxi Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/QO/C8QO00162F

Reference45 articles.

1. J. A. Joule and K.Mills , Heterocylic Chemistry , Blackwell Science, Ltd. , Oxford , 4th edn, 2000 , vol. 121

2. M. Balasubraimanan and J. G.Keay , in Comprehensive Heterocyclic Chemistry II , ed. A. R. Katritzky , C. W. Rees and E. F. V. Scriven , Pergamon Press , Oxford , 1996 , vol. 5 , p. 245

3. Quinoline, quinazoline and acridonealkaloids

4. Synthesis of brequinar analogue inhibitors of malaria parasite dihydroorotate dehydrogenase

5. Discovery of Diverse Human Dihydroorotate Dehydrogenase Inhibitors as Immunosuppressive Agents by Structure-Based Virtual Screening

Cited by 18 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Stereoselective synthesis of acyclic (Z)-3-haloallylamines via a multicomponent reaction of propargylic alcohols, TMSX and sulfonamides;Tetrahedron;2024-08

2. One-Pot Synthesis of 4-Chloroquinolines via Bis(trichloromethyl) Carbonate and Triphenylphosphine Oxide-Mediated Cascade Reactions of N-Aryl Enaminones;The Journal of Organic Chemistry;2024-07-05

3. Stereoselective Synthesis of Acyclic (Z)-3-Haloallylamines Via a Multicomponent Reaction of Propargylic Alcohols, Tmsx and Sulfonamides;2024

4. NBS-mediated bromination and dehydrogenation of tetrahydro-quinoline in one pot: scope and mechanistic study;RSC Advances;2023

5. Brønsted Acid Promoted Sulfonylation of Propargylic Alcohols: Synthesis of Triaryl Allenyl Sulfones under Mild Conditions;European Journal of Organic Chemistry;2022-12-30