Bicyclic core estrogens as full antagonists: synthesis, biological evaluation and structure–activity relationships of estrogen receptor ligands based on bridged oxabicyclic core arylsulfonamides-Reference-Cited by-同舟云学术

Bicyclic core estrogens as full antagonists: synthesis, biological evaluation and structure–activity relationships of estrogen receptor ligands based on bridged oxabicyclic core arylsulfonamides

Published:2012 Issue:43 Volume:10 Page:8692
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Zhu Manghong,Zhang Chen,Nwachukwu Jerome C.,Srinivasan Sathish,Cavett Valerie,Zheng Yangfan,Carlson Kathryn E.,Dong Chune,Katzenellenbogen John A.,Nettles Kendall W.,Zhou Hai-Bing

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2012/OB/C2OB26531A

Reference33 articles.

1. Designer Estrogens

2. Estrogen receptor transcription and transactivation Estrogen receptor alpha and estrogen receptor beta: regulation by selective estrogen receptor modulators and importance in breast cancer

3. Molecular Determinants for the Tissue Specificity of SERMs

4. Raloxifene (LY139481 HCI) prevents bone loss and reduces serum cholesterol without causing uterine hypertrophy in ovariectomized rats.

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