Trigonal scaffolds for multivalent targeting of melanocortin receptors-Reference-Cited by-同舟云学术

Trigonal scaffolds for multivalent targeting of melanocortin receptors

Published:2015 Issue:6 Volume:13 Page:1778-1791
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Elshan N. G. R. Dayan¹²³⁴,Jayasundera Thanuja⁵²³⁴,Anglin Bobbi L.¹²³⁴,Weber Craig S.⁵²³⁴,Lynch Ronald M.⁵²³⁴⁶,Mash Eugene A.¹²³⁴

Affiliation:

1. Department of Chemistry and Biochemistry

2. University of Arizona

3. Tucson

4. USA

5. Department of Physiology

6. The Bio5 Institute

Abstract

Short, efficient syntheses of multivalent molecules targeted to the human melanocortin 4 receptor based on phloroglucinol, tripropargylamine, and 1,4,7-triazacyclononane are described.

Funder

National Cancer Institute

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB02094D

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