A new cascade halosulfonylation of 1,7-enynes toward 3,4-dihydroquinolin-2(1H)-ones via sulfonyl radical-triggered addition/6-exo-dig cyclization-Reference-Cited by-同舟云学术

A new cascade halosulfonylation of 1,7-enynes toward 3,4-dihydroquinolin-2(1H)-ones via sulfonyl radical-triggered addition/6-exo-dig cyclization

Published:2016 Issue:9 Volume:52 Page:1907-1910
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Zhu Yi-Long¹²³⁴⁵,Jiang Bo¹²³⁴⁵,Hao Wen-Juan¹²³⁴⁵,Wang Ai-Fang¹²³⁴⁵,Qiu Jiang-Kai¹²³⁴⁵,Wei Ping⁶⁷⁸⁵,Wang De-Cai⁶⁷⁸⁵,Li Guigen⁹¹⁰¹¹¹²¹³,Tu Shu-Jiang¹²³⁴⁵

Affiliation:

1. School of Chemistry and Chemical Engineering

2. Jiangsu Key Laboratory of Green Synthetic Chemistry for Functional Materials

3. Jiangsu Normal University

4. Xuzhou 221116

5. P. R. China

6. Biotechnology and Pharmaceutical Engineering

7. Nanjing Tech University

8. Nanjing

9. Department of Chemistry and Biochemistry

10. Texas Tech University

11. Lubbock

12. USA

13. Institute of Chemistry & Biomedical Sciences

Abstract

A new cascade three-component halosulfonylation of 1,7-enynes for efficient synthesis of densely functionalized 3,4-dihydroquinolin-2(1H)-ones has been established from readily accessible arylsulfonyl hydrazides and NIS (or NBS).

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2016/CC/C5CC08895J

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