Redox-neutral functionalization of α-Csp3–H bonds of secondary cyclic amines: a highly atom-economical strategy for N-arylation/formal cross-dehydrogenative couplings-Reference-Cited by-同舟云学术

Redox-neutral functionalization of α-Csp3–H bonds of secondary cyclic amines: a highly atom-economical strategy for N-arylation/formal cross-dehydrogenative couplings

Published:2021 Issue:8 Volume:23 Page:2950-2955
ISSN:1463-9262
Container-title:Green Chemistry
language:en
Short-container-title:Green Chem.

Author:

Jha Priyankar¹²³⁴,Husen Saddam¹²³⁴⁵,Kumar Ravindra¹²³⁴⁵^ORCID

Affiliation:

1. Division of Medicinal and Process Chemistry

2. CSIR-Central Drug Research Institute

3. Lucknow-226031

4. India

5. Academy of Scientific & Innovative Research (AcSIR)

Abstract

An efficient redox-neutral method has been developed for α-Csp³–H functionalization of secondary cyclic amines via concurrent N-arylation/formal cross dehydrogenation coupling (CDC) with sp²-C–H and sp³-C–H bonds of arenes and ketones, respectively.

Funder

Science and Engineering Research Board

Publisher

Royal Society of Chemistry (RSC)

Subject

Pollution,Environmental Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/GC/D0GC04258G

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