Stereoselective and regioselective 5-exo-dig cyclization of 8-alkynylnaphthalen-1-amines for the synthesis of (E)-2-(arylthio)alkylene-1,2-dihydrobenzo[cd]indoles-Reference-Cited by-同舟云学术

Stereoselective and regioselective 5-exo-dig cyclization of 8-alkynylnaphthalen-1-amines for the synthesis of (E)-2-(arylthio)alkylene-1,2-dihydrobenzo[cd]indoles

Published:2018 Issue:16 Volume:16 Page:3006-3011
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Bi Cheng¹²³⁴⁵,Zhang Lianpeng¹²³⁴⁵,Qiu Guanyinsheng¹²³⁴⁵^ORCID,Li Xiaofang⁶⁷⁸⁵,Yao Jinzhong¹²³⁴⁵,Zhou Hongwei¹²³⁴⁵^ORCID

Affiliation:

1. College of Biological

2. Chemical Science and Engineering

3. Jiaxing University

4. Jiaxing 314001

5. China

6. School of Chemistry and Chemical Engineering

7. Hunan University of Science and Technology

8. Xiangtan

Abstract

A palladium and iodine-cocatalyzed 5-exo-dig aza-thiocyclization of 8-alkynylnaphthalen-1-amines for the synthesis of (E)-2-alkylene-1,2-dihydrobenzo[cd]indole thioethers is reported.

Funder

Natural Science Foundation of Zhejiang Province

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C8OB00556G

Reference51 articles.

1. Practical Methodologies for the Synthesis of Indoles

2. Recent advances in indole syntheses: New routes for a classic target