Insecticide discovery by drug repurposing: new synergistic inhibitors againstPeriplaneta americana

Author:

Chafer-Dolz Beatriz1,Cecilia José M.2,Imbernón Baldomero3,Núñez-Delicado Estrella3,Casaa-Giner Victor1,Cerón-Carrasco José P.4ORCID

Affiliation:

1. Bio Logic Crop Science, S.L. Amadeo de Saboya 1-4, 46010, Valencia, Spain

2. Universitat Politécnica de Valencia (UPV), Camino de Vera S/N, 46022, Valencia, Spain

3. Universidad Católica San Antonio de Murcia (UCAM), Campus de los Jerónimos, 30107, Murcia, Spain

4. Centro Universitario de la Defensa, Universidad Politécnica de Cartagena, C/Coronel López Peña s/n, Base Aérea de San Javier, Santiago de la Ribera, 30720, Murcia, Spain

Abstract

Virtual screening has been widely used to accelerate the drug discovery process. We adapted these methods to propose an enhanced insecticide formulation. Our numeric outcomes were confirmed by usingin vivomodels.

Funder

Ministerio de Ciencia e Innovación

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,General Chemistry,Catalysis

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