Heptadentate chelates for <sup>89</sup>Zr-radiolabelling of monoclonal antibodies-Reference-Cited by-同舟云学术

Heptadentate chelates for ⁸⁹Zr-radiolabelling of monoclonal antibodies

Published:2022 Issue:12 Volume:9 Page:3071-3081
ISSN:2052-1553
Container-title:Inorganic Chemistry Frontiers
language:en
Short-container-title:Inorg. Chem. Front.

Author:

Guillou Amaury¹^ORCID,Ouadi Ali²^ORCID,Holland Jason P.¹^ORCID

Affiliation:

1. University of Zurich, Department of Chemistry, Winterthurerstrasse 190, CH-8057, Zurich, Switzerland

2. Université de Strasbourg, CNRS, IPHC UMR 7178, F-67000, Strasbourg, France

Abstract

Herein, we report the synthesis of three new bifunctional heptadentate metal ion binding chelates derived from desferrioxamine B (DFO) linked to a tripeptide unit and photoactivatable aryl azide for conjugation to monoclonal antibodies.

Funder

Agence Nationale de la Recherche

Schweizerischer Nationalfonds zur Förderung der Wissenschaftlichen Forschung

H2020 European Research Council

Publisher

Royal Society of Chemistry (RSC)

Subject

Inorganic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/QI/D2QI00442A

Reference44 articles.

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