Rapid access to 3-acyl indoles using ethyl acetate/triflic acid couple as the acylium donor and Cu(OAc)2 catalysed aerial oxidation of indole benzoins
Author:
Affiliation:
1. Molecular Synthesis and Drug Discovery Laboratory
2. Centre of Biomedical Research
3. Sanjay Gandhi Postgraduate Institute of Medical Sciences
4. Lucknow-226014
5. India
Abstract
R′ = 1° and 2° alkyls, benzyl, allyl, cyanomethyl, carboxymethyl, phenyl; Ar = C6H5, 4-F-C6H4, 4-MeO–C6H4; X = N, O, S; Y = H, Me; Z = H, Br.
Funder
Science and Engineering Research Board
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2020/OB/D0OB01977A
Reference47 articles.
1. Esters as Acylating Reagent in a Friedel−Crafts Reaction: Indium Tribromide Catalyzed Acylation of Arenes Using Dimethylchlorosilane
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3. Enzymatic acylation: assessing the greenness of different acyl donors
4. Lipase-mediated enantioselective acylation of alcohols with functionalized vinyl esters: acyl donor tolerance and applications
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