Direct and two-step bioorthogonal probes for Bruton's tyrosine kinase based on ibrutinib: a comparative study-Reference-Cited by-同舟云学术

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Direct and two-step bioorthogonal probes for Bruton's tyrosine kinase based on ibrutinib: a comparative study

Published:2015 Issue:18 Volume:13 Page:5147-5157
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Liu Nora¹²³⁴,Hoogendoorn Sascha¹²³⁴,van de Kar Bas⁵⁶⁴,Kaptein Allard⁵⁶⁴,Barf Tjeerd⁵⁶⁴,Driessen Christoph⁷⁸⁹,Filippov Dmitri V.¹²³⁴,van der Marel Gijsbert A.¹²³⁴,van der Stelt Mario¹²³⁴,Overkleeft Herman S.¹²³⁴

Affiliation:

1. Leiden Institute of Chemistry

2. Leiden University

3. 2300 RA Leiden

4. The Netherlands

5. AcertaPharma

6. Oss

7. Kantonspital St. Gallen

8. St. Gallen

9. Switserland

Abstract

Direct and two-step activity-based probes allow for profiling of Bruton's tyrosine kinase in vitro and in situ.

Funder

European Research Council

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00474H

Reference27 articles.

1. Tec kinases: modulators of lymphocyte signaling and development

2. The role of Bruton's tyrosine kinase in B-cell development and function: a genetic perspective

3. Regulation of B Lymphocyte Development and Activation by Bruton's Tyrosine Kinase

4. Chronic active B-cell-receptor signalling in diffuse large B-cell lymphoma

5. Bruton tyrosine kinase is commonly overexpressed in mantle cell lymphoma and its attenuation by Ibrutinib induces apoptosis

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