Synthesis of N-indolated amino acids or peptides from 2-alkynylanilines via a dearomatization process-Reference-Cited by-同舟云学术

Synthesis of N-indolated amino acids or peptides from 2-alkynylanilines via a dearomatization process

Published:2021 Issue:24 Volume:8 Page:6869-6873
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Qiu Weilian¹,Wang Weiyi¹,Liu Yin²,Fan Renhua¹^ORCID

Affiliation:

1. Department of Chemistry, Fudan University, 220 Handan Road, Shanghai, 200433, China

2. Department of Breast Surgery, Fudan University Shanghai Cancer Center/Cancer Institute and Department of Oncology, Shanghai Medical College, Fudan University, Shanghai, China

Abstract

A process for the rapid synthesis of N-indolated amino acids or peptides from readily available 2-alkynylanilines via dearomatization was reported.

Funder

National Natural Science Foundation of China

Science and Technology Commission of Shanghai Municipality

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/QO/D1QO01257F

Reference36 articles.

1. Modular Total Synthesis of Protein Kinase C Activator (−)-Indolactam V

2. New Classes of Tumor Promoters: Teleocidin, Aplysiatoxin, and Palytoxin

3. Quantitative structure-activity studies on indole alkaloid tumor promoter indolactam congeners

4. Synthesis and biological activities of new conformationally fixed analogues of (−)-indolactam-V, the core structure of tumor-promoting teleocidins

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Novel chitosan-acetyl isatin polymer derivatives: synthesis, characterization, and applications in bone tissue engineering;Biomass Conversion and Biorefinery;2022-08-27

2. Synthesis of chiral N-alkylated indoles through replacement of aniline nitrogen by natural amino acids;Green Synthesis and Catalysis;2022-08

3. Divergent synthesis of 4-amino indoles with free amine groups via tandem reaction of 2-alkynylanilines;Organic Chemistry Frontiers;2022