Synthesis of bioactive and stabilized cyclic peptides by macrocyclization using C(sp3)–H activation
Author:
Affiliation:
1. State Key Laboratory of Coordination Chemistry
2. School of Chemistry and Chemical Engineering
3. Nanjing University
4. Nanjing 210093
5. China
Abstract
Synthesis of cyclic peptides with novel Cβ–Ar crosslinks has been achieved by C(sp3)–H activation, and their biological properties have been evaluated for the first time.
Funder
National Natural Science Foundation of China
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2017/SC/C6SC05530C
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